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Specific Catalysis of Asparaginyl Deamidation by Carboxylic Acids: Kinetic, Thermodynamic, and Quantitative Structure–Property Relationship Analyses

JOURNAL ARTICLE published 7 April 2014 in Molecular Pharmaceutics

Authors: Brian D. Connolly | Benjamin Tran | Jamie M. R. Moore | Vikas K. Sharma | Andrew Kosky

Rapeseed Protein-Derived Antioxidant Peptide RAP Ameliorates Nonalcoholic Steatohepatitis and Related Metabolic Disorders in Mice

JOURNAL ARTICLE published 7 January 2019 in Molecular Pharmaceutics

Research funded by Guangdong Introducing Innovative and Enterpreneurial Teams (2016ZT06Y337)

Authors: Qian Zhao | Hongjiao Xu | Sihua Hong | Nazi Song | Junqiu Xie | Zhibin Yan | Rui Wang | Pengyu Yang | Xianxing Jiang

Preclinical Evaluation of a Fluorescent Probe Targeting Receptor CDCP1 for Identification of Ovarian Cancer

JOURNAL ARTICLE published 6 September 2021 in Molecular Pharmaceutics

Research funded by National Health and Medical Research Council of Australia (APP1121970) | Tour de Cure (RSP-256-18/19) | Medical Research Future Fund (MRF1199422)

Authors: Yaowu He | Tashbib Khan | Thomas Kryza | Martina L. Jones | Justin B. Goh | Nicholas J. Lyons | Lesley A. Pearce | Michael D Lee | Madeline Gough | Rebecca Rogers | Claire M Davies | C. Blake Gilks | Thomas Hodgkinson | Rohan Lourie | Sinead C. Barry | Lewis C. Perrin | Charlotte C. Williams | Simon Puttick | Timothy E. Adams | Trent P. Munro | John D. Hooper | Naven Chetty

Drug Distribution in Microspheres Enhances Their Anti-Inflammatory Properties in the Gottingen Minipig

JOURNAL ARTICLE published 8 September 2015 in Molecular Pharmaceutics

Research funded by U.S. Department of Defense (W81XWH-07-1-0668,W81XWH-09-1-0711)

Authors: Michail Kastellorizios | Namita Tipnis | Fotios Papadimitrakopoulos | Diane J. Burgess

Targeting of Injectable Drug Nanocrystals

JOURNAL ARTICLE published 2 June 2014 in Molecular Pharmaceutics

Research funded by Swiss National Science Foundation (310030_138342)

Authors: Kathrin Fuhrmann | Marc A. Gauthier | Jean-Christophe Leroux

Genetic Targeting Strategies for Adenovirus

JOURNAL ARTICLE published 1 October 2005 in Molecular Pharmaceutics

Authors: Sam C. Noureddini | David T. Curiel

Multiple Linear Regression Modeling To Predict the Stability of Polymer–Drug Solid Dispersions: Comparison of the Effects of Polymers and Manufacturing Methods on Solid Dispersion Stability

JOURNAL ARTICLE published 7 May 2018 in Molecular Pharmaceutics

Research funded by Engineering and Physical Sciences Research Council (EP/I01375X/1)

Authors: Gudrun A. Fridgeirsdottir | Robert J. Harris | Ian L. Dryden | Peter M. Fischer | Clive J. Roberts

Isothermal Crystallization Monitoring and Time–Temperature-Transformation of Amorphous GDC-0276: Differential Scanning Calorimetric and Rheological Measurements

JOURNAL ARTICLE published 4 January 2021 in Molecular Pharmaceutics

Research funded by Division of Civil, Mechanical and Manufacturing Innovation (CMMI-1662046)

Authors: Sixue Cheng | Paroma Chakravarty | Karthik Nagapudi | Gregory B. McKenna

Standardized Preclinical In Vitro Blood–Brain Barrier Mouse Assay Validates Endocytosis-Dependent Antibody Transcytosis Using Transferrin-Receptor-Mediated Pathways

JOURNAL ARTICLE published 6 March 2023 in Molecular Pharmaceutics

Authors: Jamie I. Morrison | Alex Petrovic | Nicole G. Metzendorf | Fadi Rofo | Canan U. Yilmaz | Sofia Stenler | Hanna Laudon | Greta Hultqvist

Investigation of Deteriorated Dissolution of Amorphous Itraconazole: Description of Incompatibility with Magnesium Stearate and Possible Solutions

JOURNAL ARTICLE published 6 November 2017 in Molecular Pharmaceutics

Research funded by European Commission (FIEK 16-1-2016-0007,T?MOP 4.2.1/B-09/1/KMR-2010-0002) | Orsz?gos Tudom?nyos Kutat?si Alapprogramok (124541,K112644) | Magyarorszag Kormanya (FIEK 16-1-2016-0007,T?MOP 4.2.1/B-09/1/KMR-2010-0002)

Authors: B. Démuth | D. L. Galata | E. Szabó | B. Nagy | A. Farkas | A. Balogh | E. Hirsch | H. Pataki | Z. Rapi | L. Bezúr | T. Vigh | G. Verreck | Z. Szalay | Á. Demeter | G. Marosi | Z. K. Nagy

Characterization of Novel 18F-Labeled Phenoxymethylpyridine Derivatives as Amylin Imaging Probes

JOURNAL ARTICLE published 3 December 2018 in Molecular Pharmaceutics

Research funded by Japan Society for the Promotion of Science (14J05961,LS060)

Authors: Hiroyuki Watanabe | Masashi Yoshimura | Kohei Sano | Yoichi Shimizu | Sho Kaide | Yuji Nakamoto | Kaori Togashi | Masahiro Ono | Hideo Saji

One-Step Self-Assembling Nanomicelles for Pirarubicin Delivery To Overcome Multidrug Resistance in Breast Cancer

JOURNAL ARTICLE published 7 November 2016 in Molecular Pharmaceutics

Research funded by National Natural Science Foundation of China (81471068,81603035)

Authors: Yanping Li | Rui Li | Qinhui Liu | Wenyao Li | Ting Zhang | Min Zou | Hong Li | Tong Wu | Shihai Cheng | Zhiguang Su | Zhirong Zhang | Jinhan He

Chemical Modulation of the Human Oligopeptide Transporter 1, hPepT1

JOURNAL ARTICLE published 4 December 2017 in Molecular Pharmaceutics

Research funded by U.S. Department of Defense (W81XWH-15-1-0539) | National Institute of General Medical Sciences (R01 GM108911,R01 GM115481)

Authors: Claire Colas | Masayuki Masuda | Kazuaki Sugio | Seiji Miyauchi | Yongjun Hu | David E. Smith | Avner Schlessinger

Factors Affecting the Clearance and Biodistribution of Polymeric Nanoparticles

JOURNAL ARTICLE published 1 August 2008 in Molecular Pharmaceutics

Authors: Frank Alexis | Eric Pridgen | Linda K. Molnar | Omid C. Farokhzad

The Natural Cell-Penetrating Peptide Crotamine Targets Tumor Tissue in Vivo and Triggers a Lethal Calcium-Dependent Pathway in Cultured Cells

JOURNAL ARTICLE published 6 February 2012 in Molecular Pharmaceutics

Authors: Fabio D. Nascimento | Lucie Sancey | Alexandre Pereira | Claire Rome | Vitor Oliveira | Eduardo B. Oliveira | Helena B. Nader | Tetsuo Yamane | Irina Kerkis | Ivarne L. S. Tersariol | Jean-Luc Coll | Mirian A. F. Hayashi

The Uniqueness of Albumin as a Carrier in Nanodrug Delivery

JOURNAL ARTICLE published 3 May 2021 in Molecular Pharmaceutics

Research funded by Natural Sciences and Engineering Research Council of Canada (RGPIN-2019-05970)

Authors: Alessandra Spada | Jaber Emami | Jack A. Tuszynski | Afsaneh Lavasanifar

Differential Cytosolic Delivery and Presentation of Antigen by Listeriolysin O-Liposomes to Macrophages and Dendritic Cells

JOURNAL ARTICLE published 1 February 2005 in Molecular Pharmaceutics

Authors: Ethan M. Stier | Manas Mandal | Kyung-Dall Lee

What Are the Important Factors That Influence API Crystallization in Miscible Amorphous API–Excipient Mixtures during Long-Term Storage in the Glassy State?

JOURNAL ARTICLE published 7 February 2022 in Molecular Pharmaceutics

Authors: Ann Newman | George Zografi

Glass Transition Dynamics and Physical Stability of Amorphous Griseofulvin in Binary Mixtures with Low-Tg Excipients

JOURNAL ARTICLE published 5 August 2019 in Molecular Pharmaceutics

Research funded by Narodowe Centrum Nauki (2015/16/W/NZ7/00404)

Authors: Wenkang Tu | Justyna Knapik-Kowalczuk | Krzysztof Chmiel | Marian Paluch

Characterization of Differential Tissue Abundance of Major Non-CYP Enzymes in Human

JOURNAL ARTICLE published 2 November 2020 in Molecular Pharmaceutics

Authors: Abdul Basit | Naveen K. Neradugomma | Christopher Wolford | Peter W. Fan | Bernard Murray | Ryan H. Takahashi | S. Cyrus Khojasteh | Bill J. Smith | Scott Heyward | Rheem A. Totah | Edward J. Kelly | Bhagwat Prasad